Our offerings:
50 GPCRs in place so far, 45 stable cell lines
Class A Orphan receptors | GPR65 |
GPR68 | |
GPR84 | |
MRGPRX2 | |
MRGPRB2 (mouse ortholog) | |
GPR18, GPR55 and GPR119 | GPR119 |
Melanocortin receptors | MC1 |
MC2 | |
MC3 | |
MC4 | |
MC5 | |
5-Hydroxytryptamine receptors (Serotonin) | 5-HT1A |
5-HT2A | |
5-HT2B | |
5-HT2C | |
Acetylcholine receptors (muscarinic) | M1 |
M2 | |
Opioid receptors | MOP |
DOP | |
Orexin receptors | OX1R |
OX2R | |
Dopamine receptors | D1R |
Adenosine receptors | A2A |
Histamine receptors | H1 |
Glucagon receptor family | GLP1R |
GIPR | |
GCGR | |
GLP2R | |
mGLP1R | |
Gonadotrophin-releasing hormone receptors | GnRHR |
VIP and PACAP receptors | PAC1 (PACAP) |
Ghrelin receptor | Ghrelin/GHSR-1a |
Somatostatin receptors | SSTR2 |
Calcitonin receptors | CGRP receptor |
Free fatty acid receptors | FFA1 (GPR40) |
Bile acid receptor | GPBA receptor (TGR5) |
Chemokine receptors | CXCR1/IL-8a |
CXCR2/IL-8b | |
CXCR3 | |
CXCR4 | |
CXCR5 | |
CXCR6 | |
CX3CR1 | |
CXCR7/ACKR3 | |
Anaphylatoxin receptors (Complement peptide receptors) | C3aR |
C5aR1 | |
Apelin receptor | APJ (apelin) |
Lysophospholipid (LPA) receptors | LPA1 |